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Department of Chemistry

Han Xiao

Professor of Chemistry, Bioengineering, Biosciences

Director, SynthX Center

CPRIT Scholar in Cancer Research

The Xiao lab develops chemical biology and medicinal chemistry technologies to probe, reprogram, and treat complex biological systems, spanning cancer-targeted medicines, genetic code expansion with noncanonical amino acids, photoactivatable/NIR-II probes for deep-tissue imaging, and recent high-throughput Sequence Display approaches that integrate machine learning and protein language models to accelerate protein evolution for biomedical applications.

Public Rice profile source

Average rating

3.3

20 temporary mock ratings

Difficulty

3.5

course-linked average

Courses

9

in seeded sections

Public profile

Biography

Han Xiao is the Director of the SynthX Center and a Professor in the Departments of Chemistry, Biosciences, and Bioengineering at Rice University, where his laboratory develops chemical biology and bioengineering technologies to probe, reprogram, and treat complex biological systems. He is a CPRIT Scholar in Cancer Research and received his B.S. in Chemistry with an honors degree in physical science from the University of Science and Technology of China, completed his Ph.D. at The Scripps Research Institute with Peter G. Schultz, and completed postdoctoral training at Stanford University with Carolyn R. Bertozzi. Since launching his independent laboratory at Rice in 2017, Han has emerged as a leader in the bone delivery of therapeutics, pioneering bone-targeted biologics, antibody-drug conjugates, and immune-modulating therapies designed to concentrate treatment in the bone microenvironment; he also co-found Osteologics Therapeutics, a Curie.Bio-backed company translating this platform toward new medicines for bone metastasis and other skeletal diseases. His group is also at the forefront of Sequence Display technology, which enables unbiased, large-scale protein sequence-activity datasets that can be integrated with machine learning and protein language models to accelerate protein evolution and biomedical discovery. In parallel, he leads large-scale, multi-institutional efforts, including a recent $18 million ARPA-H award focused on advanced imaging and diagnostics for the lymphatic system. His honors include the DoD Breast Cancer Research Program Breakthrough Award (Level 2), the NIH Maximizing Investigators' Research Award, the Norman Hackerman-Welch Young Investigator Award, and the David W. Robertson Award for Excellence in Medicinal Chemistry.

Research areas

Chemical Biology, Organic Synthesis, Chemistry of Life

Keywords

Chemical biology; medicinal chemistry, machine learning; protein evolution; molecular imaging

Courses taught

BIOS 310

Ind Res For Bios Undergrads

Independent research in Rice BioSciences faculty laboratories (sections 2 and above) or other Texas Medical Center laboratories (section 1). Students must have secured a research position prior to applying for BIOS 310. Students spend at least 42 hours in the laboratory for each semester hour of credit (>9h/week for 3 credits). A minimum of 3 credit hours is needed to count toward the BS in Biosciences or to replace one required 300+ level elective lab course for the BA in Biosciences (cannot replace major concentration core labs). Requires a proposal abstract, weekly reports, and a research paper (fall/spring/summer) or a poster presentation (spring/summer for advanced students). Students wishing to perform their research in an off-campus lab must apply online (biosugresearch.rice.edu) at least 3 weeks prior to the start of classes and may not register for fewer than 3 credit hours. Students taking BIOS 310 in the full summer semester must be available to do full-time research for a minimum of 6 weeks or part-time equivalent which should equal to a total of 126 hours working in the lab. It is recommended that summer students spread their hours over 8-10 weeks. Recommended Prerequisite(s): Students are strongly advised to secure research advisors and register for the class well in advance of the start of classes. Recommended Prerequisite(s): Students are strongly advised to secure research advisors and register for the class well in advance of the start of classes. Repeatable for Credit.

BiosciencesNone1-5 credits
4.06.7hAjo-Franklin, Caroline, An, Linna, Bartel, Bonnie, Bashor, Caleb, Beason-Abmayr, Beth, Bennett, Matthew, Braam, Janet, Carson, Daniel, Catanese, Jamie, Chappell, James, de Moraes, Marcos, Dunham, Amy, Egan, Scott, Evans, Kory, Flynn, Jonathan, Gao, Yang, Glasscock, Cameron, Gustin, Michael, Hennelly, Lauren, Hilton, Isaac, Iyer, Harini, Johnson, Cassidy, Kirienko, Natasha, Kranz, Sven, Lavery, Laura, Lieberman-Aiden, Erez, Loveless, Theresa, Lu, George, Lwigale, Peter, Masiello, Carrie, Matsuda, Seiichi P., McCary, Matt, McNew, James, Miller, Thomas, Nakhleh, Luay, Nikonowicz, Edward, Novak, Joseph, Olmos, Joey, Onuchic, Jose, Rudolf, Volker, Rummel, Andrea, Segatori, Laura, Shamoo, Yousif, Siemann, Evan, Silberg, Joff, Solomon, Scott, Stewart, Charles, Tabor, Jeffrey, Tao, Yizhi, Uribe, Rosa, Wagner, Daniel, Wittung Stafshede, Pernilla, Wolynes, Peter, Xiao, Han

BIOS 401

Undergraduate Honors Research

The Biosciences Honors Research Program offers our seniors and advanced juniors the opportunity to perform a two-semester, individual research project in a research laboratory in Biosciences or an approved off-campus site and offers opportunities for students to develop their written and oral scientific communication skills. Students registering for BIOS 401 are expected to take BIOS 402 the following semester. Each semester, students are expected to average 15 hours per week in research (laboratory) and communication skills activities (scheduled through the companion seminar co-requisite). In BIOS 401, students will prepare regular progress reports, attend lab meetings, and write an end-of-semester short paper (at least 5 pages) on their work. Must register for co-requisite BIOS 411.

BiosciencesNone5 credits
3.89.8hAjo-Franklin, Caroline, An, Linna, Bartel, Bonnie, Beason-Abmayr, Beth, Bennett, Matthew, Braam, Janet, Carson, Daniel, Catanese, Jamie, Chappell, James, de Moraes, Marcos, Dunham, Amy, Egan, Scott, Evans, Kory, Gao, Yang, Gustin, Michael, Hennelly, Lauren, Kirienko, Natasha, Lavery, Laura, Lieberman-Aiden, Erez, Loveless, Theresa, Lwigale, Peter, Matsuda, Seiichi P., McCary, Matt, McNew, James, Miller, Thomas, Nakhleh, Luay, Nikonowicz, Edward, Onuchic, Jose, Rudolf, Volker, Rummel, Andrea, Segatori, Laura, Shamoo, Yousif, Siemann, Evan, Silberg, Joff, Solomon, Scott, Stewart, Charles, Tabor, Jeffrey, Tao, Yizhi, Uribe, Rosa, Wagner, Daniel, Wittung Stafshede, Pernilla, Wolynes, Peter, Xiao, Han

BIOS 611

Research Seminar

Discussion of individual research or current topics in particular areas. Intended for students conducting research projects in the lab of the instructor. Repeatable for Credit.

BiosciencesNone1 credits
3.98.2hAjo-Franklin, Caroline, An, Linna, Bartel, Bonnie, Bashor, Caleb, Bennett, Matthew, Braam, Janet, Carson, Daniel, Chappell, James, de Moraes, Marcos, Gao, Yang, Glasscock, Cameron, Gustin, Michael, Han, Yimo, Hilton, Isaac, Iyer, Harini, Kirienko, Natasha, Lavery, Laura, Lieberman-Aiden, Erez, Loveless, Theresa, Luan, Lan, Lwigale, Peter, Matsuda, Seiichi P., McNew, James, Nikonowicz, Edward, Onuchic, Jose, Rosenberg, Susan, Sawakuchi, Gabriel, Segatori, Laura, Shamoo, Yousif, Silberg, Joff, Stewart, Charles, Tao, Yizhi, Uribe, Rosa, Wagner, Daniel, Wittung Stafshede, Pernilla, Wolynes, Peter, Xiao, Han, Zhou, Zheng

BIOS 800

Bcb Graduate Research

Biochemistry & Cell Biology graduate research. Repeatable for Credit.

BiosciencesNone1-15 credits
3.96.1hAjo-Franklin, Caroline, An, Linna, Bartel, Bonnie, Bashor, Caleb, Bennett, Matthew, Braam, Janet, Carson, Daniel, Chappell, James, de Moraes, Marcos, Gao, Yang, Glasscock, Cameron, Gustin, Michael, Han, Yimo, Hilton, Isaac, Iyer, Harini, Kirienko, Natasha, Lavery, Laura, Lieberman-Aiden, Erez, Loveless, Theresa, Luan, Lan, Lwigale, Peter, Matsuda, Seiichi P., McNew, James, Nikonowicz, Edward, Onuchic, Jose, Rosenberg, Susan, Sawakuchi, Gabriel, Segatori, Laura, Shamoo, Yousif, Silberg, Joff, Stewart, Charles, Tao, Yizhi, Uribe, Rosa, Wagner, Daniel, Wittung Stafshede, Pernilla, Wolynes, Peter, Xiao, Han, Zhou, Zheng

CHEM 007

Visiting Research

Research conducted by visiting student scholars. Repeatable for Credit.

ChemistryNone0 credits
3.54.5hKolomeisky, Anatoly, Ma, Yuan, Mou, Quanbing, Renata, Hans, Sarlah, David, Shee, James, Xiao, Han, Yruegas, Samantha

CHEM 442

Medicinal Chemistry I

A course intended to provide the student with an overview of the elements of drug discover, design and development. Targets for drug discovery will be discussed, as well as considerations of drug optimization with respect to the biological target and drug metabolism. Cross-list: CHEM 542.

ChemistryNone3 credits
3.59.2hXiao, Han

CHEM 542

Medicinal Chemistry I

A course intended to provide the student with an overview of the elements of drug discover, design and development. Targets for drug discovery will be discussed, as well as considerations of drug optimization with respect to the biological target and drug metabolism. A summary of the FDA and patent processes will also be included. Cross-list: CHEM 442.

ChemistryNone3 credits
3.18.0hXiao, Han

CHEM 800

Graduate Research

Repeatable for Credit.

ChemistryNone1-15 credits
3.97.7hAjayan, Pulickel, Alvarez, Pedro, Bagchi, Kushal, Ball, Zachary, Bao, Gang, Dai, Mingjie, Diehl, Michael, Gustavsson, Anna-Karin, Hafner, Jason, Halas, Naomi, Han, Yimo, Hartgerink, Jeffrey, Hernandez Sanchez, Raul, Hulet, Randy, Igoshin, Oleg, Jones, Matt, Kampouri, Stavroula, Kolomeisky, Anatoly, Kurti, Laszlo, Lou, Jun, Ma, Yuan, MacKintosh, Frederick, Marciel, Amanda, Marti-Arbona, Angel, Martin, Lane, Masiello, Carrie, Matsuda, Seiichi P., McHugh, Kevin, Mikos, Antonios, Mohite, Aditya, Morosan, Emilia, Mou, Quanbing, Nevidomskyy, Andriy, Nienhaus, Lea, Nordlander, Peter, Onuchic, Jose, Pasquali, Matteo, Renata, Hans, Sarlah, David, Scuseria, Gustavo, Shee, James, Tour, James, Wang, Haotian, Weisman, Bruce, West, Julian, Wittung Stafshede, Pernilla, Wolynes, Peter, Wong, Michael, Xiao, Han, Yakobson, Boris, Yruegas, Samantha

SSPB 800

Graduate Research

Graduate students will conduct independent research/thesis project under the direction of their advisor. Repeatable for Credit.

Systems/Synthetic/Phys BiologyNone1-15 credits
3.35.8hAjo-Franklin, Caroline, Alvarez, Pedro, An, Linna, Bao, Gang, Bashor, Caleb, Bennett, Matthew, Butts, Jessica, Chappell, James, Dai, Mingjie, de Moraes, Marcos, Diehl, Michael, Gao, Yang, Glasscock, Cameron, Gollihar, Jimmy, Gustavsson, Anna-Karin, Hilton, Isaac, Igoshin, Oleg, Iyer, Harini, Kalluri, Raghu, Kavraki, Lydia, Kiang, Ching-Hwa, Kimmel, Marek, Kirienko, Natasha, Kolomeisky, Anatoly, Lavery, Laura, Li, Lei, Lieberman-Aiden, Erez, Loveless, Theresa, Lu, George, Luan, Lan, Ma, Yuan, MacKintosh, Frederick, Masiello, Carrie, Mou, Quanbing, Nakhleh, Luay, Nikonowicz, Edward, Onuchic, Jose, Phillips, George, Raphael, Rob, Renata, Hans, Robinson, Jacob, Segatori, Laura, Shamoo, Yousif, Silberg, Joff, St. Pierre, Francois, Stadler, Lauren, Szablowski, Jerzy, Tabor, Jeffrey, Tang, Evelyn, Tao, Yizhi, Thyer, Ross, Treangen, Todd, Uribe, Rosa, Veiseh, Omid, Vlassakis, Julea, Warmflash, Aryeh, Wolynes, Peter, Xiao, Han, Xie, Chong, Yao, Vicky

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